Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1181 |
Bradykinin (2-9)
Des-Arg1-bradykinin |
Bradykinin Receptor | GPCR/G Protein |
Bradykinin (2-9) (Des-Arg1-bradykinin),是Bradykinin的一种氨基端截短肽类代谢物,通过Aminopeptidase P的切割作用形成。 | |||
TP1999 |
MEN 11270
|
||
Peptide antagonist of the B2 bradykinin receptor (pKi = 10.3); conformationally constrained cyclized analog of HOE 140. Blocks hypotension and bronchoconstriction in vivo. Displays selectivity for B2 over 29 other receptors and ion channels (pIC50 < 5.5). |